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Amiable, C. and Paoletti, J. and Haouz, A. and Padilla, A. and Labesse, G. and Kaminski, P. A. and Pochet, S.
6-(Hetero)Arylpurine nucleotides as inhibitors of the oncogenic target DNPH1: synthesis, structural studies and cytotoxic activities
Eur J Med Chem (2014)
85, 418-37
10.1016/j.ejmech.2014.07.110
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Andre-Miral, C. and Kone, F. M. and Solleux, C. and Grandjean, C. and Dion, M. and Tran, V. and Tellier, C.
De novo design of a trans-beta-N-acetylglucosaminidase activity from a GH1 beta-glycosidase by mechanism engineering
Glycobiology (2015)
25, 394-402
10.1093/glycob/cwu121
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Angelone, T. and Caruso, A. and Rochais, C. and Caputo, A. M. and Cerra, M. C. and Dallemagne, P. and Filice, E. and Genest, D. and Pasqua, T. and Puoci, F. and Saturnino, C. and Sinicropi, M. S. and El-Kashef, H.
Indenopyrazole oxime ethers: synthesis and beta1-adrenergic blocking activity
Eur J Med Chem (2015)
92, 672-81
10.1016/j.ejmech.2015.01.037
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Antigny, F. and Norez, C. and Becq, F. and Vandebrouck, C.
CFTR and Ca Signaling in Cystic Fibrosis
Front Pharmacol (2011)
2, 67
10.3389/fphar.2011.00067
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Aouadi, W. and Blanjoie, A. and Vasseur, J. J. and Debart, F. and Canard, B. and Decroly, E.
Binding of the Methyl Donor S-Adenosyl-l-Methionine to Middle East Respiratory Syndrome Coronavirus 2'-O-Methyltransferase nsp16 Promotes Recruitment of the Allosteric Activator nsp10
J Virol (2017)
91,
10.1128/JVI.02217-16
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Aouadi, W. and Eydoux, C. and Coutard, B. and Martin, B. and Debart, F. and Vasseur, J. J. and Contreras, J. M. and Morice, C. and Querat, G. and Jung, M. L. and Canard, B. and Guillemot, J. C. and Decroly, E.
Toward the identification of viral cap-methyltransferase inhibitors by fluorescence screening assay
Antiviral Res (2017)
144, 330-339
10.1016/j.antiviral.2017.06.021
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Apel, C. and Geny, C. and Dumontet, V. and Birlirakis, N. and Roussi, F. and Pham, V. C. and Doan Thi Mai, H. and Nguyen, V. H. and Chau, V. M. and Litaudon, M.
Endiandric acid analogues from Beilschmiedia ferruginea as dual inhibitors of Bcl-xL/Bak and Mcl-1/Bid interactions
J Nat Prod (2014)
77, 1430-7
10.1021/np500170v
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Araujo, J. R. and Tomas, J. and Brenner, C. and Sansonetti, P. J.
Impact of high-fat diet on the intestinal microbiota and small intestinal physiology before and after the onset of obesity
Biochimie (2017)
141, 97-106
10.1016/j.biochi.2017.05.019
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Ardes-Guisot, N. and Alonzi, D. S. and Reinkensmeier, G. and Butters, T. D. and Norez, C. and Becq, F. and Shimada, Y. and Nakagawa, S. and Kato, A. and Bleriot, Y. and Sollogoub, M. and Vauzeilles, B.
Selection of the biological activity of DNJ neoglycoconjugates through click length variation of the side chain
Org Biomol Chem (2011)
9, 5373-88
10.1039/c1ob05119a
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Ardhaoui, M. and Bhatt, S. and Zheng, M. and Dowling, D. and Jolivalt, C. and Khonsari, F. A.
Biosensor based on laccase immobilized on plasma polymerized allylamine/carbon electrode
Mater Sci Eng C Mater Biol Appl (2013)
33, 3197-205
10.1016/j.msec.2013.03.052
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Ardhaoui, M. and Zheng, M. and Pulpytel, J. and Dowling, D. and Jolivalt, C. and Khonsari, F. A.
Plasma functionalized carbon electrode for laccase-catalyzed oxygen reduction by direct electron transfer
Bioelectrochemistry (2013)
91, 52-61
10.1016/j.bioelechem.2012.12.005
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Armando, S. and Quoyer, J. and Lukashova, V. and Maiga, A. and Percherancier, Y. and Heveker, N. and Pin, J. P. and Prezeau, L. and Bouvier, M.
The chemokine CXC4 and CC2 receptors form homo- and heterooligomers that can engage their signaling G-protein effectors and betaarrestin
FASEB J (2014)
28, 4509-23
10.1096/fj.13-242446
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Arora, R. and Di Michele, M. and Stes, E. and Vandermarliere, E. and Martens, L. and Gevaert, K. and Van Heerde, E. and Linders, J. T. and Brehmer, D. and Jacoby, E. and Bonnet, P.
Structural investigation of B-Raf paradox breaker and inducer inhibitors
J Med Chem (2015)
58, 1818-31
10.1021/jm501667n
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Assad Kahn, S. and Costa, S. L. and Gholamin, S. and Nitta, R. T. and Dubois, L. G. and Feve, M. and Zeniou, M. and Coelho, P. L. and El-Habr, E. and Cadusseau, J. and Varlet, P. and Mitra, S. S. and Devaux, B. and Kilhoffer, M. C. and Cheshier, S. H. and Moura-Neto, V. and Haiech, J. and Junier, M. P. and Chneiweiss, H.
The anti-hypertensive drug prazosin inhibits glioblastoma growth via the PKCdelta-dependent inhibition of the AKT pathway
EMBO Mol Med (2016)
8, 511-26
10.15252/emmm.201505421
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Atif, M. L. and Brenet, A. and Hageaux, S. and Fave, M. H. and Cochet, C. and Baticle, E. and Pourrier, C. and Wolny, D. and Astagneau, P. and Kadi, Z. and Standard precautions work, group
Awareness of standard precautions for 4439 healthcare professionals in 34 institutions in France
Med Mal Infect (2013)
43, 10-6
10.1016/j.medmal.2012.11.004
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Atmanene, C. and Ronin, C. and Teletchea, S. and Gautier, F. M. and Djedaini-Pilard, F. and Ciesielski, F. and Vivat, V. and Grandjean, C.
Biophysical and structural characterization of mono/di-arylated lactosamine derivatives interaction with human galectin-3
Biochem Biophys Res Commun (2017)
489, 281-286
10.1016/j.bbrc.2017.05.150
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Aubry, S. and Aubert, G. and Cresteil, T. and Crich, D.
Synthesis and biological investigation of the beta-thiolactone and beta-lactam analogs of tetrahydrolipstatin
Org Biomol Chem (2012)
10, 2629-32
10.1039/c2ob06976h
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Aubry, S. and Sasaki, K. and Eloy, L. and Aubert, G. and Retailleau, P. and Cresteil, T. and Crich, D.
Exploring the potential of the beta-thiolactones in bioorganic chemistry
Org Biomol Chem (2011)
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10.1039/c1ob05967j
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Audran, E. and Dagher, R. and Gioria, S. and Tsvetkov, P. O. and Kulikova, A. A. and Didier, B. and Villa, P. and Makarov, A. A. and Kilhoffer, M. C. and Haiech, J.
A general framework to characterize inhibitors of calmodulin: use of calmodulin inhibitors to study the interaction between calmodulin and its calmodulin binding domains
Biochim Biophys Acta (2013)
1833, 1720-31
10.1016/j.bbamcr.2013.01.008
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Aulner, N. and Danckaert, A. and Rouault-Hardoin, E. and Desrivot, J. and Helynck, O. and Commere, P. H. and Munier-Lehmann, H. and Spath, G. F. and Shorte, S. L. and Milon, G. and Prina, E.
High content analysis of primary macrophages hosting proliferating Leishmania amastigotes: application to anti-leishmanial drug discovery
PLoS Negl Trop Dis (2013)
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10.1371/journal.pntd.0002154
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Austin, S. and Taouji, S. and Chevet, E. and Wodrich, H. and Rayne, F.
Using AlphaScreen((R)) to Identify Small-Molecule Inhibitors Targeting a Conserved Host-Pathogen Interaction
Methods Mol Biol (2016)
1449, 453-67
10.1007/978-1-4939-3756-1_30
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Autelitano, F. and Loyaux, D. and Roudieres, S. and Deon, C. and Guette, F. and Fabre, P. and Ping, Q. and Wang, S. and Auvergne, R. and Badarinarayana, V. and Smith, M. and Guillemot, J. C. and Goldman, S. A. and Natesan, S. and Ferrara, P. and August, P.
Identification of novel tumor-associated cell surface sialoglycoproteins in human glioblastoma tumors using quantitative proteomics
PLoS One (2014)
9, e110316
10.1371/journal.pone.0110316
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Avarre, J. C. and Dugue, R. and Alonso, P. and Diombokho, A. and Joffrois, C. and Faivre, N. and Cochet, C. and Durand, J. D.
Analysis of the black-chinned tilapia Sarotherodon melanotheron heudelotii reproducing under a wide range of salinities: from RNA-seq to candidate genes
Mol Ecol Resour (2014)
14, 139-49
10.1111/1755-0998.12148
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Ayachi, S. and Simonin, F.
Involvement of Mammalian RF-Amide Peptides and Their Receptors in the Modulation of Nociception in Rodents
Front Endocrinol (Lausanne) (2014)
5, 158
10.3389/fendo.2014.00158
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Ayoub, M. A. and Crepieux, P. and Koglin, M. and Parmentier, M. and Pin, J. P. and Poupon, A. and Reiter, E. and Smit, M. and Steyaert, J. and Watier, H. and Wilkinson, T.
Antibodies targeting G protein-coupled receptors: Recent advances and therapeutic challenges
MAbs (2017)
9, 735-741
10.1080/19420862.2017.1325052
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Ayrolles-Torro, A. and Imberdis, T. and Torrent, J. and Toupet, K. and Baskakov, I. V. and Poncet-Montange, G. and Gregoire, C. and Roquet-Baneres, F. and Lehmann, S. and Rognan, D. and Pugniere, M. and Verdier, J. M. and Perrier, V.
Oligomeric-induced activity by thienyl pyrimidine compounds traps prion infectivity
J Neurosci (2011)
31, 14882-92
10.1523/JNEUROSCI.0547-11.2011
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Azmi, M. N. and Geny, C. and Leverrier, A. and Litaudon, M. and Dumontet, V. and Birlirakis, N. and Gueritte, F. and Leong, K. H. and Halim, S. N. and Mohamad, K. and Awang, K.
Kingianic acids A-G, Endiandric acid analogues from Endiandra kingiana
Molecules (2014)
19, 1732-47
10.3390/molecules19021732
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Bach-Segura, P. and Belarbi, N.
[Diagnostic imaging evaluation of neonatal vomiting]
J Radiol (2011)
92, 134-41
10.1016/j.jradio.2010.12.007
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Baddour-Hadjean, R. and Boudaoud, A. and Bach, S. and Emery, N. and Pereira-Ramos, J. P.
A comparative insight of potassium vanadates as positive electrode materials for Li batteries: influence of the long-range and local structure
Inorg Chem (2014)
53, 1764-72
10.1021/ic402897d
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Baklouti, A. and Goulet, A. and Lichiere, J. and Canard, B. and Charrel, R. N. and Ferron, F. and Coutard, B. and Papageorgiou, N.
Toscana virus nucleoprotein oligomer organization observed in solution
Acta Crystallogr D Struct Biol (2017)
73, 650-659
10.1107/S2059798317008774
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Ballereau, S. and Levade, T. and Genisson, Y. and Andrieu-Abadie, N.
Alteration of ceramide 1-O-functionalization as a promising approach for cancer therapy
Anticancer Agents Med Chem (2012)
12, 316-28
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Baratte, B. and Serive, B. and Bach, S.
[Screening marine resources to find novel chemical inhibitors of disease-relevant protein kinases]
Med Sci (Paris) (2015)
31, 538-45
10.1051/medsci/20153105016
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Barbier, J. and Cintrat, J. C. and Gillet, D.
Intracellular pathogens convert macrophages from death traps into hospitable homes
FEBS J (2016)
283, 595-7
10.1111/febs.13657
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Barelier, S. and Krimm, I.
Ligand specificity, privileged substructures and protein druggability from fragment-based screening
Curr Opin Chem Biol (2011)
15, 469-74
10.1016/j.cbpa.2011.02.020
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Barelier, S. and Linard, D. and Pons, J. and Clippe, A. and Knoops, B. and Lancelin, J. M. and Krimm, I.
Discovery of fragment molecules that bind the human peroxiredoxin 5 active site
PLoS One (2010)
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Barelier, S. and Pons, J. and Gehring, K. and Lancelin, J. M. and Krimm, I.
Ligand specificity in fragment-based drug design
J Med Chem (2010)
53, 5256-66
10.1021/jm100496j
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Barelier, S. and Pons, J. and Marcillat, O. and Lancelin, J. M. and Krimm, I.
Fragment-based deconstruction of Bcl-xL inhibitors
J Med Chem (2010)
53, 2577-88
10.1021/jm100009z
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[Strength and specificity of the CMBA screening platform for bioactive molecules discovery]
Med Sci (Paris) (2015)
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10.1051/medsci/20153104017
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Barral, K. and Priet, S. and De Michelis, C. and Sire, J. and Neyts, J. and Balzarini, J. and Canard, B. and Alvarez, K.
Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates
Eur J Med Chem (2010)
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10.1016/j.ejmech.2009.11.012
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Development of specific dengue virus 2'-O- and N7-methyltransferase assays for antiviral drug screening
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Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication
Eur J Med Chem (2011)
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Barthe, P. and Veyron-Churlet, R. and de Visch, A. and Gilleron, M. and Saliou, J. M. and Tomavo, S. and Nigou, J. and Brodin, P. and Cohen-Gonsaud, M.
Mycobacterium tuberculosis LppM Displays an Original Structure and Domain Composition Linked to a Dual Localization
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The One-Class Classification Approach to Data Description and to Models Applicability Domain
Mol Inform (2010)
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2P2Idb: a structural database dedicated to orthosteric modulation of protein-protein interactions
Nucleic Acids Res (2013)
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Electronic, spectroscopic, and ion-sensing properties of a dehydro[m]pyrido[14]- and [15]annulene isomer library
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A strategy to discover decoy chemokine ligands with an anti-inflammatory activity
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Fragment-based discovery of a new family of non-peptidic small-molecule cyclophilin inhibitors with potent antiviral activities
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Vasohibins/SVBP are tubulin carboxypeptidases (TCPs) that regulate neuron differentiation
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Mitochondrial protein sorting as a therapeutic target for ATP synthase disorders
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Palladium-Catalyzed Chemoselective and Biocompatible Functionalization of Cysteine-Containing Molecules at Room Temperature
Chemistry (2016)
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Alabdul Magid, A. and Morjani, H. and Harakat, D. and Madoulet, C. and Dumontet, V. and Lavaud, C.
Triterpenoid glycosides from the leaves of Meliosma henryi
Phytochemistry (2015)
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Enzalutamide induced acute generalized exanthematous pustulosis
J Dermatol Case Rep (2016)
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Structural basis for selective recognition of acyl chains by the membrane-associated acyltransferase PatA
Nat Commun (2016)
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