Amiable, C. and Paoletti, J. and Haouz, A. and Padilla, A. and Labesse, G. and Kaminski, P. A. and Pochet, S.

6-(Hetero)Arylpurine nucleotides as inhibitors of the oncogenic target DNPH1: synthesis, structural studies and cytotoxic activities

Eur J Med Chem (2014)

85, 418-37

10.1016/j.ejmech.2014.07.110

Andre-Miral, C. and Kone, F. M. and Solleux, C. and Grandjean, C. and Dion, M. and Tran, V. and Tellier, C.

De novo design of a trans-beta-N-acetylglucosaminidase activity from a GH1 beta-glycosidase by mechanism engineering

Glycobiology (2015)

25, 394-402

10.1093/glycob/cwu121

Angelone, T. and Caruso, A. and Rochais, C. and Caputo, A. M. and Cerra, M. C. and Dallemagne, P. and Filice, E. and Genest, D. and Pasqua, T. and Puoci, F. and Saturnino, C. and Sinicropi, M. S. and El-Kashef, H.

Indenopyrazole oxime ethers: synthesis and beta1-adrenergic blocking activity

Eur J Med Chem (2015)

92, 672-81

10.1016/j.ejmech.2015.01.037

Antigny, F. and Norez, C. and Becq, F. and Vandebrouck, C.

CFTR and Ca Signaling in Cystic Fibrosis

Front Pharmacol (2011)

2, 67

10.3389/fphar.2011.00067

Aouadi, W. and Blanjoie, A. and Vasseur, J. J. and Debart, F. and Canard, B. and Decroly, E.

Binding of the Methyl Donor S-Adenosyl-l-Methionine to Middle East Respiratory Syndrome Coronavirus 2'-O-Methyltransferase nsp16 Promotes Recruitment of the Allosteric Activator nsp10

J Virol (2017)

91,

10.1128/JVI.02217-16

Aouadi, W. and Eydoux, C. and Coutard, B. and Martin, B. and Debart, F. and Vasseur, J. J. and Contreras, J. M. and Morice, C. and Querat, G. and Jung, M. L. and Canard, B. and Guillemot, J. C. and Decroly, E.

Toward the identification of viral cap-methyltransferase inhibitors by fluorescence screening assay

Antiviral Res (2017)

144, 330-339

10.1016/j.antiviral.2017.06.021

Apel, C. and Geny, C. and Dumontet, V. and Birlirakis, N. and Roussi, F. and Pham, V. C. and Doan Thi Mai, H. and Nguyen, V. H. and Chau, V. M. and Litaudon, M.

Endiandric acid analogues from Beilschmiedia ferruginea as dual inhibitors of Bcl-xL/Bak and Mcl-1/Bid interactions

J Nat Prod (2014)

77, 1430-7

10.1021/np500170v

Araujo, J. R. and Tomas, J. and Brenner, C. and Sansonetti, P. J.

Impact of high-fat diet on the intestinal microbiota and small intestinal physiology before and after the onset of obesity

Biochimie (2017)

141, 97-106

10.1016/j.biochi.2017.05.019

Ardes-Guisot, N. and Alonzi, D. S. and Reinkensmeier, G. and Butters, T. D. and Norez, C. and Becq, F. and Shimada, Y. and Nakagawa, S. and Kato, A. and Bleriot, Y. and Sollogoub, M. and Vauzeilles, B.

Selection of the biological activity of DNJ neoglycoconjugates through click length variation of the side chain

Org Biomol Chem (2011)

9, 5373-88

10.1039/c1ob05119a

Ardhaoui, M. and Bhatt, S. and Zheng, M. and Dowling, D. and Jolivalt, C. and Khonsari, F. A.

Biosensor based on laccase immobilized on plasma polymerized allylamine/carbon electrode

Mater Sci Eng C Mater Biol Appl (2013)

33, 3197-205

10.1016/j.msec.2013.03.052

Ardhaoui, M. and Zheng, M. and Pulpytel, J. and Dowling, D. and Jolivalt, C. and Khonsari, F. A.

Plasma functionalized carbon electrode for laccase-catalyzed oxygen reduction by direct electron transfer

Bioelectrochemistry (2013)

91, 52-61

10.1016/j.bioelechem.2012.12.005

Armando, S. and Quoyer, J. and Lukashova, V. and Maiga, A. and Percherancier, Y. and Heveker, N. and Pin, J. P. and Prezeau, L. and Bouvier, M.

The chemokine CXC4 and CC2 receptors form homo- and heterooligomers that can engage their signaling G-protein effectors and betaarrestin

FASEB J (2014)

28, 4509-23

10.1096/fj.13-242446

Arora, R. and Di Michele, M. and Stes, E. and Vandermarliere, E. and Martens, L. and Gevaert, K. and Van Heerde, E. and Linders, J. T. and Brehmer, D. and Jacoby, E. and Bonnet, P.

Structural investigation of B-Raf paradox breaker and inducer inhibitors

J Med Chem (2015)

58, 1818-31

10.1021/jm501667n

Assad Kahn, S. and Costa, S. L. and Gholamin, S. and Nitta, R. T. and Dubois, L. G. and Feve, M. and Zeniou, M. and Coelho, P. L. and El-Habr, E. and Cadusseau, J. and Varlet, P. and Mitra, S. S. and Devaux, B. and Kilhoffer, M. C. and Cheshier, S. H. and Moura-Neto, V. and Haiech, J. and Junier, M. P. and Chneiweiss, H.

The anti-hypertensive drug prazosin inhibits glioblastoma growth via the PKCdelta-dependent inhibition of the AKT pathway

EMBO Mol Med (2016)

8, 511-26

10.15252/emmm.201505421

Atif, M. L. and Brenet, A. and Hageaux, S. and Fave, M. H. and Cochet, C. and Baticle, E. and Pourrier, C. and Wolny, D. and Astagneau, P. and Kadi, Z. and Standard precautions work, group

Awareness of standard precautions for 4439 healthcare professionals in 34 institutions in France

Med Mal Infect (2013)

43, 10-6

10.1016/j.medmal.2012.11.004

Atmanene, C. and Ronin, C. and Teletchea, S. and Gautier, F. M. and Djedaini-Pilard, F. and Ciesielski, F. and Vivat, V. and Grandjean, C.

Biophysical and structural characterization of mono/di-arylated lactosamine derivatives interaction with human galectin-3

Biochem Biophys Res Commun (2017)

489, 281-286

10.1016/j.bbrc.2017.05.150

Aubry, S. and Aubert, G. and Cresteil, T. and Crich, D.

Synthesis and biological investigation of the beta-thiolactone and beta-lactam analogs of tetrahydrolipstatin

Org Biomol Chem (2012)

10, 2629-32

10.1039/c2ob06976h

Aubry, S. and Sasaki, K. and Eloy, L. and Aubert, G. and Retailleau, P. and Cresteil, T. and Crich, D.

Exploring the potential of the beta-thiolactones in bioorganic chemistry

Org Biomol Chem (2011)

9, 7134-43

10.1039/c1ob05967j

Audran, E. and Dagher, R. and Gioria, S. and Tsvetkov, P. O. and Kulikova, A. A. and Didier, B. and Villa, P. and Makarov, A. A. and Kilhoffer, M. C. and Haiech, J.

A general framework to characterize inhibitors of calmodulin: use of calmodulin inhibitors to study the interaction between calmodulin and its calmodulin binding domains

Biochim Biophys Acta (2013)

1833, 1720-31

10.1016/j.bbamcr.2013.01.008

Aulner, N. and Danckaert, A. and Rouault-Hardoin, E. and Desrivot, J. and Helynck, O. and Commere, P. H. and Munier-Lehmann, H. and Spath, G. F. and Shorte, S. L. and Milon, G. and Prina, E.

High content analysis of primary macrophages hosting proliferating Leishmania amastigotes: application to anti-leishmanial drug discovery

PLoS Negl Trop Dis (2013)

7, e2154

10.1371/journal.pntd.0002154

Austin, S. and Taouji, S. and Chevet, E. and Wodrich, H. and Rayne, F.

Using AlphaScreen((R)) to Identify Small-Molecule Inhibitors Targeting a Conserved Host-Pathogen Interaction

Methods Mol Biol (2016)

1449, 453-67

10.1007/978-1-4939-3756-1_30

Autelitano, F. and Loyaux, D. and Roudieres, S. and Deon, C. and Guette, F. and Fabre, P. and Ping, Q. and Wang, S. and Auvergne, R. and Badarinarayana, V. and Smith, M. and Guillemot, J. C. and Goldman, S. A. and Natesan, S. and Ferrara, P. and August, P.

Identification of novel tumor-associated cell surface sialoglycoproteins in human glioblastoma tumors using quantitative proteomics

PLoS One (2014)

9, e110316

10.1371/journal.pone.0110316

Avarre, J. C. and Dugue, R. and Alonso, P. and Diombokho, A. and Joffrois, C. and Faivre, N. and Cochet, C. and Durand, J. D.

Analysis of the black-chinned tilapia Sarotherodon melanotheron heudelotii reproducing under a wide range of salinities: from RNA-seq to candidate genes

Mol Ecol Resour (2014)

14, 139-49

10.1111/1755-0998.12148

Ayachi, S. and Simonin, F.

Involvement of Mammalian RF-Amide Peptides and Their Receptors in the Modulation of Nociception in Rodents

Front Endocrinol (Lausanne) (2014)

5, 158

10.3389/fendo.2014.00158

Ayoub, M. A. and Crepieux, P. and Koglin, M. and Parmentier, M. and Pin, J. P. and Poupon, A. and Reiter, E. and Smit, M. and Steyaert, J. and Watier, H. and Wilkinson, T.

Antibodies targeting G protein-coupled receptors: Recent advances and therapeutic challenges

MAbs (2017)

9, 735-741

10.1080/19420862.2017.1325052

Ayrolles-Torro, A. and Imberdis, T. and Torrent, J. and Toupet, K. and Baskakov, I. V. and Poncet-Montange, G. and Gregoire, C. and Roquet-Baneres, F. and Lehmann, S. and Rognan, D. and Pugniere, M. and Verdier, J. M. and Perrier, V.

Oligomeric-induced activity by thienyl pyrimidine compounds traps prion infectivity

J Neurosci (2011)

31, 14882-92

10.1523/JNEUROSCI.0547-11.2011

Azmi, M. N. and Geny, C. and Leverrier, A. and Litaudon, M. and Dumontet, V. and Birlirakis, N. and Gueritte, F. and Leong, K. H. and Halim, S. N. and Mohamad, K. and Awang, K.

Kingianic acids A-G, Endiandric acid analogues from Endiandra kingiana

Molecules (2014)

19, 1732-47

10.3390/molecules19021732

Bach-Segura, P. and Belarbi, N.

[Diagnostic imaging evaluation of neonatal vomiting]

J Radiol (2011)

92, 134-41

10.1016/j.jradio.2010.12.007

Baddour-Hadjean, R. and Boudaoud, A. and Bach, S. and Emery, N. and Pereira-Ramos, J. P.

A comparative insight of potassium vanadates as positive electrode materials for Li batteries: influence of the long-range and local structure

Inorg Chem (2014)

53, 1764-72

10.1021/ic402897d

Baklouti, A. and Goulet, A. and Lichiere, J. and Canard, B. and Charrel, R. N. and Ferron, F. and Coutard, B. and Papageorgiou, N.

Toscana virus nucleoprotein oligomer organization observed in solution

Acta Crystallogr D Struct Biol (2017)

73, 650-659

10.1107/S2059798317008774

Ballereau, S. and Levade, T. and Genisson, Y. and Andrieu-Abadie, N.

Alteration of ceramide 1-O-functionalization as a promising approach for cancer therapy

Anticancer Agents Med Chem (2012)

12, 316-28

Baratte, B. and Serive, B. and Bach, S.

[Screening marine resources to find novel chemical inhibitors of disease-relevant protein kinases]

Med Sci (Paris) (2015)

31, 538-45

10.1051/medsci/20153105016

Barbier, J. and Cintrat, J. C. and Gillet, D.

Intracellular pathogens convert macrophages from death traps into hospitable homes

FEBS J (2016)

283, 595-7

10.1111/febs.13657

Barelier, S. and Krimm, I.

Ligand specificity, privileged substructures and protein druggability from fragment-based screening

Curr Opin Chem Biol (2011)

15, 469-74

10.1016/j.cbpa.2011.02.020

Barelier, S. and Linard, D. and Pons, J. and Clippe, A. and Knoops, B. and Lancelin, J. M. and Krimm, I.

Discovery of fragment molecules that bind the human peroxiredoxin 5 active site

PLoS One (2010)

5, e9744

10.1371/journal.pone.0009744

Barelier, S. and Pons, J. and Gehring, K. and Lancelin, J. M. and Krimm, I.

Ligand specificity in fragment-based drug design

J Med Chem (2010)

53, 5256-66

10.1021/jm100496j

Barelier, S. and Pons, J. and Marcillat, O. and Lancelin, J. M. and Krimm, I.

Fragment-based deconstruction of Bcl-xL inhibitors

J Med Chem (2010)

53, 2577-88

10.1021/jm100009z

Barette, C. and Soleilhac, E. and Charavay, C. and Cochet, C. and Fauvarque, M. O.

[Strength and specificity of the CMBA screening platform for bioactive molecules discovery]

Med Sci (Paris) (2015)

31, 423-31

10.1051/medsci/20153104017

Barral, K. and Priet, S. and De Michelis, C. and Sire, J. and Neyts, J. and Balzarini, J. and Canard, B. and Alvarez, K.

Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates

Eur J Med Chem (2010)

45, 849-56

10.1016/j.ejmech.2009.11.012

Barral, K. and Sallamand, C. and Petzold, C. and Coutard, B. and Collet, A. and Thillier, Y. and Zimmermann, J. and Vasseur, J. J. and Canard, B. and Rohayem, J. and Debart, F. and Decroly, E.

Development of specific dengue virus 2'-O- and N7-methyltransferase assays for antiviral drug screening

Antiviral Res (2013)

99, 292-300

10.1016/j.antiviral.2013.06.001

Barral, K. and Weck, C. and Payrot, N. and Roux, L. and Durafour, C. and Zoulim, F. and Neyts, J. and Balzarini, J. and Canard, B. and Priet, S. and Alvarez, K.

Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication

Eur J Med Chem (2011)

46, 4281-8

10.1016/j.ejmech.2011.06.034

Barthe, P. and Veyron-Churlet, R. and de Visch, A. and Gilleron, M. and Saliou, J. M. and Tomavo, S. and Nigou, J. and Brodin, P. and Cohen-Gonsaud, M.

Mycobacterium tuberculosis LppM Displays an Original Structure and Domain Composition Linked to a Dual Localization

Structure (2016)

24, 1788-1794

10.1016/j.str.2016.07.009

Baskin, II and Kireeva, N. and Varnek, A.

The One-Class Classification Approach to Data Description and to Models Applicability Domain

Mol Inform (2010)

29, 581-7

10.1002/minf.201000063

Baskin, II and Solov'ev, V. P. and Bagatur'yants, A. A. and Varnek, A.

Predictive cartography of metal binders using generative topographic mapping

J Comput Aided Mol Des (2017)

31, 701-714

10.1007/s10822-017-0033-6

Basse, M. J. and Betzi, S. and Bourgeas, R. and Bouzidi, S. and Chetrit, B. and Hamon, V. and Morelli, X. and Roche, P.

2P2Idb: a structural database dedicated to orthosteric modulation of protein-protein interactions

Nucleic Acids Res (2013)

41, D824-7

10.1093/nar/gks1002

Basse, M. J. and Betzi, S. and Morelli, X. and Roche, P.

2P2Idb v2: update of a structural database dedicated to orthosteric modulation of protein-protein interactions

Database (Oxford) (2016)

2016,

10.1093/database/baw007

Baxter, P. N. and Al Ouahabi, A. and Gisselbrecht, J. P. and Brelot, L. and Varnek, A.

Electronic, spectroscopic, and ion-sensing properties of a dehydro[m]pyrido[14]- and [15]annulene isomer library

J Org Chem (2012)

77, 126-42

10.1021/jo201595s

Abboud, D. and Daubeuf, F. and Do, Q. T. and Utard, V. and Villa, P. and Haiech, J. and Bonnet, D. and Hibert, M. and Bernard, P. and Galzi, J. L. and Frossard, N.

A strategy to discover decoy chemokine ligands with an anti-inflammatory activity

Sci Rep (2015)

5, 14746

10.1038/srep14746

Abdelkafi, H. and Cintrat, J. C.

Regioselective Halogenation of 1,4-Benzodiazepinones via CH Activation

Sci Rep (2015)

5, 12131

10.1038/srep12131

Abdelkafi, H. and Michau, A. and Clerget, A. and Buisson, D. A. and Johannes, L. and Gillet, D. and Barbier, J. and Cintrat, J. C.

Synthesis, Chiral Separation, Absolute Configuration Assignment, and Biological Activity of Enantiomers of Retro-1 as Potent Inhibitors of Shiga Toxin

ChemMedChem (2015)

10, 1153-6

10.1002/cmdc.201500139